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Nuclear Receptor Compounds

Inhibitors and modulators are available for a wide range of nuclear receptor targets.

Finding Your Compound: browse through the target categories below or use the Search Box above. Still can't find what you're looking for - contact us directly at sales@mayflowerbio.com and we'll work to source it for you through our extensive supplier network.

Nuclear Receptor Categories

Androgen Receptor

Estrogen Receptors

Glucocorticoid Receptor

Liver X Receptor-like Receptors

Mineralocorticoid Receptor

Nerve Growth Factor IB-like Receptors

Peroxisome Proliferator-activated Receptors

Progesterone Receptor

Retinoic Acid Receptors

Retinoid X Receptors

Thyroid Hormone Receptors

Vitamin D Receptor-like Receptors

 


Androgen Receptor

2-Hydroxyflutamide (AR antagonist)

Bicalutamide (AR antagonist)

R-Bicalutamide (AR antagonist)

Canrenone (Na+/K+ ATPase partial agonist, aldosterone and AR antagonist)

Chlormadinone Acetate (AR and ER antagonist)

Cimetidine (Histamine H2 and AR antagonist, catalase inhibitor)

Cyproterone Acetate (AR antagonist)

Danazol (weak AR agonist)

Flutamide (AR antagonist)

Gestrinone (AR agonist, ER and PR antagonist)

Imazalil (14-α demethylase and aromatase inhibitor, AR antagonist)

Medroxyprogesterone 17-Acetate (PR, AR, glucocorticoid agonist, 3α-hydroxysteroid dehydrogenase inhibitor)

Minoxidil (AR antagonist)

Spironolactone (AR antagonist, ENaC channel blocker, potential voltage-gated Ca2+ channel blocker)

Tibolone (SERM, PR and AR agonist, aromatase inhibitor, glucocorticoid and mineralocorticoid antagonist)

Toremifene Base (SERM, androgen modulator)

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Estrogen Receptors

(E)-4-Hydroxytamoxifen (SERM modulator)

(E,Z)-4-Hydroxytamoxifen (SERM modulator)

(Z)-4-Hydroxytamoxifen (SERM modulator)

17-α-Ethynylestradiol (ER agonist)

17α-Hydroxyprogesterone Caproate (ER antagonist)

Alternariol (topoisomerase I and II inhibitor, potential ER agonist)

Alternariol-9-methyl Ether (oxidative phosphorylation inhibitor, potential ER agonist)

Bakuchiol (ERα agonist)

Clomiphene Citrate (FIASMA, SERM)

Coumestrol (ERβ agonist, aromatase and 3α-hydroxysteroid dehydrogenase inhibitor)

Dehydroepiandrosterone (ERβ, NMDA, σ1 agonist, ERα and AR partial agonist, GABA-A antagonist)

Diethylstilbestrol (ER agonist)

Droloxifene (SERM modulator)

Droloxifene Citrate (SERM modulator)

(±)-Equol (ER agonist)

Estradiol (ER agonist)

Estriol (ER agonist)

Estrone (ER agonist)

Genistin (SERM modulator)

Gestrinone (AR agonist, ER and PR antagonist)

Hexestrol (ER agonist, microtubule polymerization inhibitor)

Naringin (SERM modulator)

Quinestrol (ER agonist)

Raloxifene Hydrochloride (SERM modulator)

Tamoxifen Citrate (FIASMA, SERM, PKC inhibitor)

Tibolone (SERM, PR and AR agonist, aromatase inhibitor, glucocorticoid and mineralocorticoid antagonist)

Toremifene Base (SERM, androgen modulator)

Zearalenone (ER agonist)

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Glucocorticoid Receptor

Betamethasone (glucocorticoid agonist)

Betamethasone 21-Phosphate Sodium (glucocorticoid agonist)

Betamethasone Valerate (glucocorticoid agonist)

Budesonide (glucocorticoid agonist)

Clobetasol Propionate (glucocorticoid agonist)

Deflazacort (Oxazoline; glucocorticoid agonist)

Dexamethasone (Glucocorticoid agonist)

Dexamethasone Acetate Monohydrate (glucocorticoid agonist)

Dexamethasone Phosphate Sodium (glucocorticoid agonist)

Fluocinolone Acetonide (glucocorticoid agonist)

Hydrocortisone (glucocorticoid agonist)

Hydrocortisone 21-Acetate (glucocorticoid agonist)

Medroxyprogesterone 17-Acetate (PR, AR, glucocorticoid agonist, 3α-hydroxysteroid dehydrogenase inhibitor)

Methylprednisolone (glucocorticoid agonist)

Miconazole (14-α demethylase inhibitor, potential glucocorticoid antagonist)

Miconazole Nitrate (14-α demethylase inhibitor, potential glucocorticoid antagonist)

Mifepristone (PR and glucocorticoid antagonist)

Prednisolone (glucocorticoid agonist)

Prednisolone Sodium Phosphate (glucocorticoid agonist)

Prednisone (glucocorticoid agonist)

Prednisone Acetate (glucocorticoid agonist)

Tibolone (SERM, PR and AR agonist, aromatase inhibitor, glucocorticoid and mineralocorticoid antagonist)

Triamcinolone (glucocorticoid agonist)

Triamcinolone Acetonide (glucocorticoid agonist)

Triamcinolone Acetonide Acetate (glucocorticoid agonist)

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Liver X Receptor-like Receptors

Cafestol (FXR and PXR agonist, ERK2 and MEK1 inhibitor)

Cafestol Acetate (FXR and PXR agonist, ERK2 and MEK1 inhibitor)

Cafestol Eicosanate (FXR and PXR agonist, ERK2 and MEK1 inhibitor)

Cafestol Linoleate (FXR and PXR agonist, ERK2 and MEK1 inhibitor)

Cafestol Oleate (FXR and PXR agonist, ERK2 and MEK1 inhibitor)

Cafestol Palmitate (FXR and PXR agonist, ERK2 and MEK1 inhibitor)

Cafestol Stearate (FXR and PXR agonist, ERK2 and MEK1 inhibitor)

Chenodeoxycholic Acid (FXR agonist)

Guggulsterone (FXR antagonist)

Vesicular Stomatitis Virus Peptide (LDLR agonist)

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Mineralocorticoid Receptor

α-Melanocyte Stimulating Hormone (MCR agonist)

[Nle4, D-Phe7]-α-Melanocyte Stimulating Hormone (MCR agonist)

β-Melanocyte Stimulating Hormone, human (MCR agonist)

γ-1 Melanocyte Stimulating Hormone (MCR agonist)

γ-3 Melanocyte Stimulating Hormone (MCR agonist)

Melanotan II (MCR agonist)

Progesterone (PR agonist, mineralocorticoid, nAChR, σ1/2 antagonist)

Tibolone (SERM, PR and AR agonist, aromatase inhibitor, glucocorticoid and mineralocorticoid antagonist)

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Nerve Growth Factor IB-like Receptors

Tuftsin (Nrp1 agonist)

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Peroxisome Proliferator-activated Receptors

5-Aminosalicylic Acid (PPARγ agonist, potential COX-1/2 inhibitor)

5-Methoxyindole (potential PPARγ and 5-HT3 agonist)

Auraptene (PPARα agonist, ACAT inhibitor)

Azelaic Acid (PPARγ agonist, KLK5 inhibitor)

Bezafibrate (PPARα agonist)

Biochanin A (potential PPARα and PPARγ agonist)

Ciglitazone (PPARγ agonist)

Ciprofibrate (PPARα agonist)

Clofibrate (PPARα agonist)

Clofibric Acid (PPARα agonist)

Fenofibrate (PPARα agonist)

Gemfibrozil (PPARα agonist, enoyl-CoA reductase inhibitor)

Ginsenoside Re (PPARγ agonist)

Irbesartan (PPARγ agonist, AT1 inhibitor)

γ-Linolenic Acid (6c, 9c, 12c) (PPAR agonist)

Mycophenolic Acid (PPARγ agonist, IMPDH inhibitor, microtubule polymerization inhibitor)

Phytanic Acid (RXR and PPAR agonist, potential GPR40 agonist)

Pioglitazone Hydrochloride (PPARα/γ agonist, mitoNEET modulator)

Pseudoginsenoside F11 (PPARγ agonist)

Rosiglitazone (PPARγ agonist)

Rosiglitazone Maleate (PPARγ agonist)

Shogaol (PPARγ agonist, 5-HT3 antagonist)

Telmisartan (AT-II antagonist, PPARγ/δ modulator)

Triflumizole (PPARγ agonist, RORγ inverse agonist, 14-α demethylase and aromatase inhibitor, ubiquitin/proteasome modulator)

Troglitazone (PPARγ agonist, ATP-sensitive K+ channel blocker)

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Progesterone Receptor

Altrenogest (PR agonist)

Ethisterone (PR agonist)

Gestrinone (AR agonist, ER and PR antagonist)

Medroxyprogesterone 17-Acetate (PR, AR, glucocorticoid agonist, 3α-hydroxysteroid dehydrogenase inhibitor)

Mifepristone (PR and glucocorticoid antagonist)

Norethindrone (PR agonist)

Progesterone (PR agonist, mineralocorticoid, nAChR, σ1/2 antagonist)

Stanozolol (PR agonist)

Tibolone (SERM, PR and AR agonist, aromatase inhibitor, glucocorticoid and mineralocorticoid antagonist)

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Retinoic Acid Receptors

Acitretin (RARα/β/γ agonist)

Adapalene (RARα/β/γ agonist)

all-trans-Retinol (RAR and RXR agonist)

all-trans-Retinol, high purity (RAR/RXR agonist)

Etretinate (RAR, RXR agonist)

Lycopene (RAR agonist)

Tamibarotene (RARα/β agonist)

9-cis-Retinoic Acid (RAR and RXR agonist)

13-cis-Retinoic Acid (RAR and RXR agonist)

trans-Retinoic Acid (RAR agonist)

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Retinoid X Receptors

Bexarotene (RXR agonist)

Etretinate (RAR, RXR agonist)

Phytanic Acid (RXR and PPAR agonist, potential GPR40 agonist)

9-cis-Retinoic Acid (RAR and RXR agonist)

13-cis-Retinoic Acid (RAR and RXR agonist)

all-trans-Retinol (RAR and RXR agonist)

all-trans-Retinol, high purity (RAR/RXR agonist)

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Thyroid Hormone Receptors

L-Thyroxine Sodium Pentahydrate (Endogenous thyroid hormone T4)

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Vitamin D Receptor-like Receptors

25-Hydroxyvitamin D2 (VDR agonist)

25-Hydroxyvitamin D3 (VDR agonist)

Cafestol (FXR and PXR agonist, ERK2 and MEK1 inhibitor)

Cafestol Acetate (FXR and PXR agonist, ERK2 and MEK1 inhibitor)

Cafestol Eicosanate (FXR and PXR agonist, ERK2 and MEK1 inhibitor)

Cafestol Linoleate (FXR and PXR agonist, ERK2 and MEK1 inhibitor)

Cafestol Oleate (FXR and PXR agonist, ERK2 and MEK1 inhibitor)

Cafestol Palmitate (FXR and PXR agonist, ERK2 and MEK1 inhibitor)

Cafestol Stearate (FXR and PXR agonist, ERK2 and MEK1 inhibitor)

Calcitriol (VDR agonist)

Ginkgolide A (GSK-3β inhibitor, potential PXR agonist)

Guggulsterone (FXR antagonist)

LCL-161 (PXR agonist, IAP inhibitor)

Strontium Ranelate (potential CaR agonist)

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